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Publications 2017

(148)     Pereira, M. D. F.; Sarghe, E.; Rouillard, H.; Domon, L.; Chrouvrier, J.-R.; Thiry, V. Synthesis of Novel Heterocyclic Fused Pyrimidin-4-One Derivatives from Imino-1,2,3-Dithiazoles. Arkivoc 2017, 2017, 335–345.
doi : 10.24820/ark.5550190.p010.256.

(147)     Di Poi, C.; Costil, K.; Bouchart, V.; Halm-Lemeille, M.-P. Toxicity Assessment of Five Emerging Pollutants, Alone and in Binary or Ternary Mixtures, towards Three Aquatic Organisms. Environ. Sci. Pollut. Res. 2017.
doi : 10.1007/s11356-017-9306-9.

(146)     Fogha, J.; Marekha, B.; De Giorgi, M.; Voisin-Chiret, A. S.; Rault, S.; Bureau, R.; Sopkova-De Oliveira Santos, J. Toward Understanding Mcl-1 Promiscuous and Specific Binding Mode. J. Chem. Inf. Model. 2017, 57, 2885–2895.
doi : 10.1021/acs.jcim.7b00396.

(145)     Rabatel, J.; Fannes, T.; Lepailleur, A.; Le Goff, J.; Crémilleux, B.; Ramon, J.; Bureau, R.; Cuissart, B. Non a Priori Automatic Discovery of 3D Chemical Patterns: Application to Mutagenicity. Mol. Inform. 2017, 36, 1700022.
doi : 10.1002/minf.201700022.

(144)     Leprince, J.; Bagnol, D.; Bureau, R.; Fukusumi, S.; Granata, R.; Hinuma, S.; Larhammar, D.; Primeaux, S.; Sopkova-de Oliveiras Santos, J.; Tsutsui, K.; Ukena, K.; Vaudry, H. The Arg-Phe-Amide Peptide 26RFa/glutamine RF-Amide Peptide and Its Receptor: IUPHAR Review 24. Br. J. Pharmacol. 2017, 174, 3573–3607.
doi: 10.1111/bph.13907

(143)     Kieffer, C.; Babin, V.; Jouanne, M.; Slimani, I.; Berhault, Y.; Legay, R.; Sopková-de Oliveira Santos, J.; Rault, S.; Voisin-Chiret, A. S. Sequential One Pot Double C H Heteroarylation of Thiophene Using Bromopyridines to Synthesize Unsymmetrical 2,5-Bipyridylthiophenes. Tetrahedron 2017, 73, 5509–5516.
doi: 10.1016/j.tet.2017.07.049

(142)     Sapi, J.; Van Hijfte, L.; Dallemagne, P. The 52 Nd International Conference on Medicinal Chemistry (RICT 2016) of the French Medicinal Chemistry Society (SCT) Held in Caen (Normandy). ChemMedChem 2017, 12, 862–871.
doi: 10.1002/cmdc.201700336

(141)     Jouanne, M.; Rault, S.; Voisin-Chiret, A.-S. Tau Protein Aggregation in Alzheimer’s Disease: An Attractive Target for the Development of Novel Therapeutic Agents. Eur. J. Med. Chem. 2017, 139, 153–167.
doi: 10.1016/j.ejmech.2017.07.070

(140)     Peauger, L.; Azzouz, R.; Gembus, V.; Tîntas, M.-L.; Sopková-de Oliveira Santos, J.; Bohn, P.; Papamicaël, C.; Levacher, V. Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation. J. Med. Chem. 2017, 60, 5909–5926.
doi: 10.1021/acs.jmedchem.7b00702

(139)   Jourdan, J.-P.; Since, M.; El Kihel, L.; Lecoutey, C.; Corvaisier, S.; Legay, R.; Sopkova-de Oliveira Santos, J.; Cresteil, T.; Malzert-Fréon, A.; Rochais, C.; Dallemagne, P. Benzylphenylpyrrolizinones with Anti-Amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer’s Disease Treatment. ChemMedChem 2017, 12, 913–916.
doi: 10.1002/cmdc.201700102.
(138)     Lalut, J.; Karila, D.; Dallemagne, P.; Rochais, C. Modulating 5-HT 4 and 5-HT 6 Receptors in Alzheimer’s Disease Treatment. Future Med. Chem. 2017, 9, 781–795.
doi : 10.4155/fmc-2017-0031


(137)     Ugarte, W.; Boizumault, P.; Crémilleux, B.; Lepailleur, A.; Loudni, S.; Plantevit, M.; Raïssi, C.; Soulet, A. Skypattern Mining: From Pattern Condensed Representations to Dynamic Constraint Satisfaction Problems. Artif. Intell. 2017, 244, 48–69.
doi: 10.1016/j.artint.2015.04.003

(136)     Haensele, E.; Mele, N.; Miljak, M.; Read, C. M.; Whitley, D. C.; Banting, L.; Delépée, C.; Sopkova-de Oliveira Santos, J.; Lepailleur, A.; Bureau, R.; Essex, J. W.; Clark, T. Conformation and Dynamics of Human Urotensin II and Urotensin Related Peptide in Aqueous Solution. J. Chem. Inf. Model. 2017, 57, 298–310.
doi : 10.1021/acs.jcim.6b00706

(135)     Poezevara, G.; Lozano, S.; Cuissart, B.; Bureau, R.; Bureau, P.; Croixmarie, V.; Vayer, P.; Lepailleur, A. A Computational Selection of Metabolite Biomarkers Using Emerging Pattern Mining: A Case Study in Human Hepatocellular Carcinoma. J. Proteome Res. 2017, 16, 2240–2249.
doi: 10.1021/acs.jproteome.7b00054

(134)     Groo, A.-C.; De Pascale, M.; Voisin-Chiret, A.-S.; Corvaisier, S.; Since, M.; Malzert-Fréon, A. Comparison of 2 Strategies to Enhance Pyridoclax Solubility: Nanoemulsion Delivery System versus Salt Synthesis. Eur. J. Pharm. Sci. 2017, 97, 218–226.
doi: 10.1016/j.ejps.2016.11.025

(133)     Iacopetta, D.; Rosano, C.; Puoci, F.; Parisi, O. I.; Saturnino, C.; Caruso, A.; Longo, P.; Ceramella, J.; Malzert-Fréon, A.; Dallemagne, P.; Rault, S.; Sinicropi, M. S. Multifaceted Properties of 1,4-Dimethylcarbazoles: Focus on Trimethoxybenzamide and Trimethoxyphenylurea Derivatives as Novel Human Topoisomerase II Inhibitors. Eur. J. Pharm. Sci. 2017, 96, 263–272.
doi : 10.1016/j.ejps.2016.09.039

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Dernière modification : 3 juillet 2020



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