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Publications 2014

(101)    Villain, J.; Lozano, S.; Halm-Lemeille, M.-P.; Durrieu, G.; Bureau, R. Quantile Regression Model for a Diverse Set of Chemicals: Application to Acute Toxicity for Green Algae. J. Mol. Model. 2014, 20, 2508.

(100)    Ursuegui, S.; Chivot, N.; Moutin, S.; Burr, A.; Fossey, C.; Cailly, T.; Laayoun, A.; Fabis, F.; Laurent, A. Biotin-Conjugated N-Methylisatoic Anhydride: A Chemical Tool for Nucleic Acid Separation by Selective 2’-Hydroxyl Acylation of RNA. Chem. Commun. 2014, 50, 5748–5751.

(99)    Rezg, R.; Mornagui, B.; Santos, J. S. O.; Dulin, F.; El-Fazaa, S.; El-haj, N. Ben; Bureau, R.; Gharbi, N. Protective Effects of Caffeic Acid against Hypothalamic Neuropeptides Alterations Induced by Malathion in Rat. Environ. Sci. Pollut. Res. 2014, 22, 6198–6207.

(98)    Primas, N.; Suzanne, P.; Verhaeghe, P.; Hutter, S.; Kieffer, C.; Laget, M.; Cohen, A.; Broggi, J.; Lancelot, J.-C.; Lesnard, A.; Dallemagne, P.; Rathelot, P.; Rault, S.; Vanelle, P.; Azas, N. Synthesis and in Vitro Evaluation of 4-trichloromethylpyrrolo[1,2-A]quinoxalines as New Antiplasmodial Agents. Eur. J. Med. Chem. 2014, 83, 26–35.

(97)    Péron, F.; Fossey, C.; Sopkova-Deoliveirasantos, J.; Cailly, T.; Fabis, F. Room-Temperature Ortho-Alkoxylation and -Halogenation of N-Tosylbenzamides by Using palladium(II)-Catalyzed C-H Activation. Chem. - A Eur. J. 2014, 20, 7507–7513.

(96)         Perato, S.; Giorgi, M.; Burzicki, G.; Legalite, F.; Rault, S.; Voisin-Chiret, A. Focus on Microwaves Assisted Halogen-Halogen Exchange Reaction Conditions on 2-Halopyridines. Curr. Microw. Chem. 2014, 1, 75–80.

(95)    Panno, A.; Sinicropi, M. S.; Caruso, A.; El-Kashef, H.; Lancelot, J.-C.; Aubert, G.; Lesnard, A.; Cresteil, T.; Rault, S. New Trimethoxybenzamides and Trimethoxyphenylureas Derived from Dimethylcarbazole as Cytotoxic Agents. Part I. J. Heterocycl. Chem. 2014, 51, E294–E302.

(94)    Neveu, C.; Dulin, F.; Lefranc, B.; Galas, L.; Calbrix, C.; Bureau, R.; Rault, S.; Chuquet, J.; Boutin, J. a; Guilhaudis, L.; Ségalas-Milazzo, I.; Vaudry, D.; Vaudry, H.; Santos, J. S. O.; Leprince, J. Molecular Basis of Agonist Docking in a Human GPR103 Homology Model by Site-Directed Mutagenesis and Structure-Activity Relationship Studies. Br. J. Pharmacol. 2014, 171, 4425–4439.

(93)    Minguez, L.; Pedelucq, J.; Farcy, E.; Ballandonne, C.; Budzinski, H.; Halm-Lemeille, M.-P. Toxicities of 48 Pharmaceuticals and Their Freshwater and Marine Environmental Assessment in Northwestern France. Environ. Sci. Pollut. Res. 2014.

(92)    Minguez, L.; Halm-Lemeille, M. P.; Costil, K.; Bureau, R.; Lebel, J. M.; Serpentini, A. Assessment of Cytotoxic and Immunomodulatory Properties of Four Antidepressants on Primary Cultures of Abalone Hemocytes (Haliotis Tuberculata). Aquat. Toxicol. 2014, 153, 3–11.

(91)    Minguez, L.; Farcy, E.; Ballandonne, C.; Lepailleur, A.; Serpentini, A.; Lebel, J. M.; Bureau, R.; Halm-Lemeille, M. P. Acute Toxicity of 8 Antidepressants: What Are Their Modes of Action? Chemosphere 2014, 108, 314–319.

(90)    Minguez, L.; Di Poi, C.; Farcy, E.; Ballandonne, C.; Benchouala, A.; Bojic, C.; Cossu-Leguille, C.; Costil, K.; Serpentini, A.; Lebel, J.-M.; Halm-Lemeille, M.-P. Comparison of the Sensitivity of Seven Marine and Freshwater Bioassays as Regards Antidepressant Toxicity Assessment. Ecotoxicology 2014, 23, 1744–1754.

(89)    Letullier, A.; Minguez, L.; Costil, K.; Halm-Lemeille, M.-P.; Lebel, J.-M.; Serpentini, A. In Vitro Effect of Five Pharmaceuticals on the Viability of the European Abalone Hemocytes, Haliotis Tuberculata. J. Xenobiotics 2014, 4, 78–80.

(88)    Lepailleur, A.; Freret, T.; Lemaître, S.; Boulouard, M.; Dauphin, F.; Hinschberger, A.; Dulin, F.; Lesnard, A.; Bureau, R.; Rault, S. Dual Histamine H3R/serotonin 5-HT4R Ligands with Antiamnesic Properties: Pharmacophore-Based Virtual Screening and Polypharmacology. J. Chem. Inf. Model. 2014, 54, 1773–1784.

(87)    Lepailleur, A.; Bureau, R.; Halm-Lemeille, M.-P.; Bouquet, M.; Pecquet, R.; Paris-Soubayrol, C.; Goff, J. L.; André, V.; Lecluse, Y.; Lebailly, P.; Maire, M.-A.; Vasseur, P. Assessment of the Genotoxic and Carcinogenic Potentials of 3-Aminothiophene Derivatives Using in Vitro and in Silico Methodologies. J. Appl. Toxicol. 2014, 34, 775–786.

(86)    Lecoutey, C.; Hedou, D.; Freret, T.; Giannoni, P.; Gaven, F.; Since, M.; Bouet, V.; Ballandonne, C.; Corvaisier, S.; Malzert Fréon, A.; Mignani, S.; Cresteil, T.; Boulouard, M.; Claeysen, S.; Rochais, C.; Dallemagne, P. Design of Donecopride, a Dual Serotonin Subtype 4 Receptor Agonist/acetylcholinesterase Inhibitor with Potential Interest for Alzheimer’s Disease Treatment. Proc. Natl. Acad. Sci. U. S. A. 2014, 111, E3825–E3830.

(85)    Halm-Lemeille, M. P.; Abbaszadeh Fard, E.; Latire, T.; Ferard, J. F.; Costil, K.; Lebel, J. M.; Bureau, R.; Serpentini, A. The Effect of Different Polychlorinated Biphenyls on Two Aquatic Models, the Green Alga Pseudokirchneriella Subcapitata and the Haemocytes from the European Abalone Haliotis Tuberculata. Chemosphere 2014, 110, 120–128.

(84)    Fontaine, F.; Hequet, A.; Voisin-Chiret, A. S.; Bouillon, A.; Lesnard, A.; Cresteil, T.; Jolivalt, C.; Rault, S. First Identification of Boronic Species as Novel Potential Inhibitors of the Staphylococcus Aureus NorA Efflux Pump. J. Med. Chem. 2014, 57, 2536–2548.

(83)    Dumas, N.; Moulin-Sallanon, M.; Ginovart, N.; Tournier, B. B.; Suzanne, P.; Cailly, T.; Fabis, F.; Rault, S.; Charnay, Y.; Millet, P. Small-Animal Single-Photon Emission Computed Tomographic Imaging of the Brain Serotoninergic Systems in Wild-Type and Mdr1a Knockout Rats. Mol. Imaging 2014, 13, 1–12.

(82)    Dulin, F.; Zatylny-Gaudin, C.; Ballandonne, C.; Guillet, B.; Bonafos, R.; Bureau, R.; Halm, M. P. Protecting Honey Bees: Identification of a New Varroacide by in Silico, in Vitro, and in Vivo Studies. Parasitol. Res. 2014, 113, 4601–4610.

(81)    Dubost, E.; Stiebing, S.; Ferrary, T.; Cailly, T.; Fabis, F.; Collot, V. A General Synthesis of Diversely Substituted Indazoles and Hetero-Aromatic Derivatives from O-Halo-(het)arylaldehydes or -Phenones. Tetrahedron 2014, 70, 8413–8418.

(80)    Caruso, A.; Stefania, M.; Lancelot, J.; El-kashef, H.; Saturnino, C.; Aubert, G.; Ballandonne, C.; Lesnard, A.; Cresteil, T.; Dallemagne, P.; Rault, S. Synthesis and Evaluation of Cytotoxic Activities of New Guanidines Derived from Carbazoles. Bioorg. Med. Chem. Lett. 2014, 24, 467–472.

(79)    Caruso, A.; Lancelot, J.-C.; El-Kashef, H.; Panno, A.; Sinicropi, M. S.; Legay, R.; Lesnard, A.; Lepailleur, A.; Rault, S. Four Partners, Three-Step, One-Pot Reaction for a Library of New 2-Alkyl(dialkyl)aminoquinazolin-4(3 H )-Ones. J. Heterocycl. Chem. 2014, 51, E282–E293.

(78)    Brossard, D.; Lechevrel, M.; El Kihel, L.; Quesnelle, C.; Khalid, M.; Moslemi, S.; Reimund, J.-M. Synthesis and Biological Evaluation of Bile Carboxamide Derivatives with pro-Apoptotic Effect on Human Colon Adenocarcinoma Cell Lines. Eur. J. Med. Chem. 2014, 86, 279–290.

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Dernière modification : 13 septembre 2015



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