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Publications 2012

(57)    Voisin-Chiret, A. S.; Rault, S. Using Halo (het) Arylboronic Species to Achieve Synthesis of Foldamers as Protein–protein Interaction Disruptors. Pure Appl. Chem. 2012, 84, 2467–2478.

(56)    Voisin-Chiret, A. S.; Burzicki, G.; Perato, S.; De Giorgi, M.; Franchini, C.; Sopková-De Oliveira Santos, J.; Rault, S. Aromatic Garlands, as New Foldamers, to Mimic Protein Secondary Structure. Tetrahedron 2012, 68, 4381–4389.

(55)    Villemin, D.; Cheikh, N.; Liao, L.; Bar, N.; Lohier, J. F.; Sopkova, J.; Choukchou-Braham, N.; Mostefa-Kara, B. Two Versatile Routes towards Cerpegin and Analogues: Applications of a One Pot Reaction to New Analogues of Cerpegin. Tetrahedron 2012, 68, 4906–4918.

(54)    Sopkova-De Oliveira Santos, J.; Voisin-Chiret, A. S.; Burzicki, G.; Sebaoun, L.; Sebban, M.; Lohier, J. F.; Legay, R.; Oulyadi, H.; Bureau, R.; Rault, S. Structural Characterizations of Oligopyridyl Foldamers, α-Helix Mimetics. In Journal of Chemical Information and Modeling; 2012; Vol. 52, pp. 429–439.

(53)    Primas, N.; Verhaeghe, P.; Cohen, A.; Kieffer, C.; Dumètre, A.; Hutter, S.; Rault, S.; Rathelot, P.; Azas, N.; Vanelle, P. A New Synthetic Route to Original Sulfonamide Derivatives in 2-Trichloromethylquinazoline Series: A Structure-Activity Relationship Study of Antiplasmodial Activity. Molecules 2012, 17, 8105–8117.

(52)    Péron, F.; Fossey, C.; Cailly, T.; Fabis, F. N-Tosylcarboxamide as a Transformable Directing Group for Pd-Catalyzed C-H Ortho-Arylation. Org. Lett. 2012, 14, 1827–1829.

(51)    Perato, S.; Voisin-Chiret, A. S.; Sopková-De Oliveira Santos, J.; Legay, R.; Oulyadi, H.; Rault, S. Synthesis of New Linear Poly(phenylpyridyl) Chains. Tetrahedron 2012, 68, 1910–1917.

(50)    Paloque, L.; Verhaeghe, P.; Casanova, M.; Castera-Ducros, C.; Dumètre, A.; Mbatchi, L.; Hutter, S.; Kraiem-M’Rabet, M.; Laget, M.; Remusat, V.; Rault, S.; Rathelot, P.; Azas, N.; Vanelle, P. Discovery of a New Antileishmanial Hit in 8-Nitroquinoline Series. Eur. J. Med. Chem. 2012, 54, 75–86.

(49)    Lohou, E.; Sopkova-De Oliveira Santos, J.; Schumann-Bard, P.; Boulouard, M.; Stiebing, S.; Rault, S.; Collot, V. New Hypotheses for the Binding Mode of 4- and 7-Substituted Indazoles in the Active Site of Neuronal Nitric Oxide Synthase. Bioorganic Med. Chem. 2012, 20, 5296–5304.

(48)    Lecoutey, C.; Rochais, C.; Genest, D.; Butt-Gueulle, S.; Ballandonne, C.; Corvaisier, S.; Dulin, F.; Lepailleur, A.; Sopkova-de Oliveira Santos, J.; Dallemagne, P. Synthesis of Dual AChE/5-HT4 Receptor Multi-Target Directed Ligands. MedChemComm, 2012, 3, 627–634.

(47)    Kihel, L. El. Oxidative Metabolism of Dehydroepiandrosterone (DHEA) and Biologically Active Oxygenated Metabolites of DHEA and Epiandrosterone (EpiA) - Recent Reports. Steroids, 2012, 77, 10–26.

(46)    Freret, T.; Bouet, V.; Quiedeville, A.; Nee, G.; Dallemagne, P.; Rochais, C.; Boulouard, M. Synergistic Effect of Acetylcholinesterase Inhibition (donepezil) and 5-HT(4) Receptor Activation (RS67333) on Object Recognition in Mice. Behav. Brain Res. 2012, 230, 304–308.

(45)    Dulin, F.; Halm-Lemeille, M. P.; Lozano, S.; Lepailleur, A.; Sopkova-de Oliveira Santos, J.; Rault, S.; Bureau, R. Interpretation of Honeybees Contact Toxicity Associated to Acetylcholinesterase Inhibitors. Ecotoxicol. Environ. Saf. 2012, 79, 13–21.

(44)    Dubost, E.; Dumas, N.; Fossey, C.; Magnelli, R.; Butt-Gueulle, S.; Ballandonne, C.; Caignard, D. H.; Dulin, F.; Sopkova De-Oliveira Santos, J.; Millet, P.; Charnay, Y.; Rault, S.; Cailly, T.; Fabis, F. Synthesis and Structure-Affinity Relationships of Selective High-Affinity 5-HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers. J. Med. Chem. 2012, 55, 9693–9707.

(43)    De Fatima Pereira, M.; Thiéry, V. One-Pot Synthesis of pyrrolo[1,2-A]quinoxaline Derivatives via Iron-Promoted Aryl Nitro Reduction and Aerobic Oxidation of Alcohols. Org. Lett. 2012, 14, 4754–4757.

(42)    Chosson, E.; Santoro, F.; Rochais, C.; Santos, J. S. O.; Legay, R.; Thoret, S.; Cresteil, T.; Sinicropi, M. S.; Besson, T.; Dallemagne, P. Synthesis of Novel 7-Oxo and 7-Hydroxy Trifluoroallocolchicinoids with Cytotoxic Effect. Bioorg. Med. Chem. 2012, 20, 2614–2623.

(41)    Caruso, A.; Chimento, A.; El-Kashef, H.; Lancelot, J.-C.; Panno, A.; Pezzi, V.; Saturnino, C.; Sinicropi, M. S.; Sirianni, R.; Rault, S. Antiproliferative Activity of Some 1,4-Dimethylcarbazoles on Cells That Express Estrogen Receptors: Part I. Journal of Enzyme Inhibition and Medicinal Chemistry, 2012, 27, 609–613.

(40)    Bruel, A.; Logé, C.; Tauzia, M. L. De; Ravache, M.; Le Guevel, R.; Guillouzo, C.; Lohier, J. F.; Oliveira Santos, J. S. De; Lozach, O.; Meijer, L.; Ruchaud, S.; Bénédetti, H.; Robert, J. M. Synthesis and Biological Evaluation of New 5-Benzylated 4-Oxo-3,4-Dihydro-5H-pyridazino[4,5-B]indoles as PI3Kα Inhibitors. Eur. J. Med. Chem. 2012, 57, 225–233.

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Dernière modification : 13 septembre 2015



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