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Publications 2011

(39)    Verhaeghe, P.; Dumètre, A.; Castera-Ducros, C.; Hutter, S.; Laget, M.; Fersing, C.; Prieri, M.; Yzombard, J.; Sifredi, F.; Rault, S.; Rathelot, P.; Vanelle, P.; Azas, N. 4-Thiophenoxy-2-Trichloromethyquinazolines Display in Vitro Selective Antiplasmodial Activity against the Human Malaria Parasite Plasmodium Falciparum. Bioorg. Med. Chem. Lett. 2011, 21, 6003–6006.

(38)    Rochais, C.; Yougnia, R.; Cailly, T.; Sopková-de Oliveira Santos, J.; Rault, S.; Dallemagne, P. One-Pot Synthesis of New Aza- and Diaza-Aminophenanthrenes. Tetrahedron 2011, 67, 5806–5810.

(37)    Marassio, G.; Prangé, T.; David, H. N.; Santos, J. S. O.; Gabison, L.; Delcroix, N.; Abraini, J. H.; Colloc’h, N. Pressure-Response Analysis of Anesthetic Gases Xenon and Nitrous Oxide on Urate Oxidase: A Crystallographic Study. FASEB J. 2011, 25, 2266–2275.

(36)    Lohou, E.; Collot, V.; Stiebing, S.; Rault, S. Direct Access to 3-Aminoindazoles by Buchwald-Hartwig C-N Coupling Reaction. Synthesis (Stuttg). 2011, 2651–2663.

(35)    Lecoutey, C.; Fossey, C.; Rault, S.; Fabis, F. Efficient Room-Temperature One-Pot Synthesis of 2-Amino-3-alkyl(3-Aryl)quinazolin-4(3H)-Ones. European J. Org. Chem. 2011, 2011, 2785–2788.

(34)    Julienne, D.; Delacroix, O.; Lohier, J.-F.; de Oliveira-Santos, J. S.; Gaumont, A.-C. Mechanistic Insights into the Palladium-Catalysed Asymmetric Phosphination of Cyclohexenyl Triflate (Eur. J. Inorg. Chem. 16/2011). Eur. J. Inorg. Chem. 2011, 2489–2554.

(33)    Guillot, M. V.; Desforges, A. S.; Voisin-Chiret, A. S.; Schumann, P.; Launay, A.; Lecomte, C. 296 Evaluating the Use of Megestrol Acetate in Caen and Lisieux CF Centers (2007–2010). J. Cyst. Fibros. 2011, 10, S75.

(32)    Gautier, B.; Miteva, M. A.; Goncalves, V.; Huguenot, F.; Coric, P.; Bouaziz, S.; Seijo, B.; Gaucher, J. F.; Broutin, I.; Garbay, C.; Lesnard, A.; Rault, S.; Inguimbert, N.; Villoutreix, B. O.; Vidal, M. Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by in Silico and in Vitro Screening. Chem. Biol. 2011, 18, 1631–1639.

(31)    Dubost, E.; Fossey, C.; Cailly, T.; Rault, S.; Fabis, F. Selective Ortho -Bromination of Substituted Benzaldoximes Using Pd-Catalyzed C-H Activation: Application to the Synthesis of Substituted 2-Bromobenzaldehydes. J. Org. Chem. 2011, 76, 6414–6420.

(30)    De Giorgi, M.; Voisin-Chiret, A. S.; Sopková-De Oliveira Santos, J.; Corbo, F.; Franchini, C.; Rault, S. Design and Synthesis of Thienylpyridyl Garlands as Non-Peptidic Alpha Helix Mimetics and Potential Protein-Protein Interactions Disruptors. Tetrahedron 2011, 67, 6145–6154.

(29)    Chosson, E.; Rochais, C.; Legay, R.; Sopkova de Oliveira Santos, J.; Rault, S.; Dallemagne, P. First and Mild Synthesis of Fluorene-9-Malonic Acid and Some Substituted Derivatives via the Intramolecular Hydroarylation of 2-Phenylbenzylidenemalonic Acids. Tetrahedron 2011, 67, 2548–2554.

(28)    Cheikh, N.; Bar, N.; Choukchou-Braham, N.; Mostefa-Kara, B.; Lohier, J. F.; Sopkova, J.; Villemin, D. Efficient Synthesis of New Butenolides by Subsequent Reactions: Application for the Synthesis of Original Iminolactones, Bis-Iminolactones and Bis-Lactones. Tetrahedron 2011, 67, 1540–1551.

(27)    Castera-Ducros, C.; Azas, N.; Verhaeghe, P.; Hutter, S.; Garrigue, P.; Dumtre, A.; Mbatchi, L.; Laget, M.; Remusat, V.; Sifredi, F.; Rault, S.; Rathelot, P.; Vanelle, P. Targeting the Human Malaria Parasite Plasmodium Falciparum: In Vitro Identification of a New Antiplasmodial Hit in 4-Phenoxy-2- Trichloromethylquinazoline Series. Eur. J. Med. Chem. 2011, 46, 4184–4191.

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Dernière modification : 13 septembre 2015



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